Երկիր: Թայվան
Լեզու: չինարեն
Աղբյուրը: 衛生福利部食品藥物管理署 (Ministry of Health and Welfare, Food And Drug Administration)
SITAGLIPTIN (AS MONOHYDRATE PHOSPHATE SALT)
美商默沙東藥廠股份有限公司台灣分公司 台北市信義區信義路五段106號12樓 (86683720)
A10BH01
膜衣錠
SITAGLIPTIN (AS MONOHYDRATE PHOSPHATE SALT) (9200088510) (eq. to sitagliptin 25 mg)MG
鋁箔盒裝
製 劑
須由醫師處方使用
MERCK SHARP & DOHME LTD. SHOTTON LANE, CRAMLINGTON, NORTHUMBERLAND, NE23 3JU, UNITED KINGDOM GB
sitagliptin
第二型糖尿病。
註銷日期: 2016/08/15; 註銷理由: 自請註銷; 有效日期: 2017/07/13; 英文品名: JANUVIA 25 mg F.C. Tablets
已註銷
2007-07-13
JANUVIA ( ) JANUVIA JANUVIA ( ) JANUVIA JANUVIA JANUVIA JANUVIA JANUVIA ESRD JANUVIA ( ) JANUVIA JANUVIA ( metformin 33$5Ȗ thiazolidinedione) JANUVIA JANUVIA sulfonylurea ( ) sulfonylurea ( ) JANUVIA Stevens-Johnson syndrome JANUVIA JANUVIA ( ) 250 mg/kg 125 mg/kg ( 100 mg/day 32 22 ) sitagliptin 1000 mg/kg/day ( 100 mg/day 100 ) ( ) 1000 mg/kg/day JANUVIA JANUVIA Sitagliptin sitagliptin JANUVIA JANUVIA 18 ) ) JANUVIA ( ) JANUVIA 32.13 128.5 sitagliptin phosphate monohydrate 25 50 100 JANUVIA microcrystalline cellulose anhydrous dibasic calcium phosphate (calcium hydrogen phosphate, anhydrous) croscarmellose sodium magnesium stearate sodium stearyl fumarate polyvinyl alcohol polyethylene glycol (macrogol) talc titanium dioxide red iron oxide yellow iron oxide JANUVIA (sitagliptin phosphate) GLSHSWLG\OSHSWLGDVH '33 '33 (incretin) '33 sitagliptin -1 (glucagonlike peptide-1 GLP-1) (glucose-dependent insulinotropic polypeptide GIP) Incretins GLP-1 GIP ȕ (insulin) GLP-1 Į (glucagon) sulfonylureas sulfonylureas sulfonylurea Sitagliptin '33 DPP-8 DPP-9 Sitagliptin GLP-1 sulfonylureas meglitinides biguanides (peroxisome proliferator-activated receptor gamma 33$5Ȗ Į amylin JANUVIA 100 metformin sulfonylurea ( metformin) 33$5Ȗ ( thiazolidinedione) metformin sulfonylurea metformin 33$5Ȗ JANUVIA JANUVIA sulfonylurea sulfonylurea ( ) ( >&U&O@P/PLQ PJG/ PJG/ JANUVIA &U&O <50 mL/min ! PJG/ >1.5 PJG/ JANUVIA 50 (CrCl<30 mL/min >3.0 mg/dL >2.5 mg/dL) (ESRD) JANUVIA 25 JANUVIA JANUVIA Sitagliptin &<3$ 2C8 2C9 ' 1A2 2C19 % CYP &<3$ Sitagliptin P (p-glycoprotein) P digoxin sitagliptin Sitagliptin - Sitagliptin ( ) sitagliptin metformin glyburide simvastatin rosiglitazone warfarin &<3$ CYP2C8 CYP2C9 (OCT) sitagliptin digoxin _Metformin: _ sitagliptin metformin (OCT ) metformin sitagliptin OCT _Sulfonylureas: _ sitagliptin glyburide (CYP2C9 ) glyburide CYP2C9 sulfonylurea ( glipizide tolbutamide glimepiride) _Simvastatin: _ sitagliptin VLPYDVWDWLQ Կարդացեք ամբողջական փաստաթուղթը